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-Structure paper
Title | Azepanone-based inhibitors of human and rat cathepsin K |
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Journal, issue, pages | J. Med. Chem., Vol. 44, Page 1380-1395, Year 2001 |
Publish date | Jan 6, 2003 (structure data deposition date) |
Authors | Marquis, R.W. / Ru, Y. / LoCastro, S.M. / Zeng, J. / Yamashita, D.S. / Oh, H.J. / Erhard, K.F. / Davis, L.D. / Tomaszek, T.A. / Tew, D. ...Marquis, R.W. / Ru, Y. / LoCastro, S.M. / Zeng, J. / Yamashita, D.S. / Oh, H.J. / Erhard, K.F. / Davis, L.D. / Tomaszek, T.A. / Tew, D. / Salyers, K. / Proksch, J. / Ward, K. / Smith, B. / Levy, M. / Cummings, M.D. / Haltiwanger, R.C. / Trescher, G. / Wang, B. / Hemling, M.E. / Quinn, C.J. / Cheng, H.-Y. / Lin, F. / Smith, W.W. / Janson, C.A. / Zhao, B. / McQueney, M.S. / D'Alessio, K. / Lee, C.P. / Marzulli, A. / A Dodds, R. / Blake, S. / Hwang, S.M. / James, I.E. / Gress, C.J. / Bradley, B.R. / Lark, M.W. / Gowen, M. / Veber, D.F. |
External links | J. Med. Chem. / PubMed:11311061 |
Methods | X-ray diffraction |
Resolution | 2.4 - 2.8 Å |
Structure data | PDB-1nl6: PDB-1nlj: |
Chemicals | ChemComp-750: ChemComp-2CA: |
Source |
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Keywords | HYDROLASE / SULFHYDRYL PROTEINASE |