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-Structure paper
Title | X-ray structure of human stromelysin catalytic domain complexed with nonpeptide inhibitors: implications for inhibitor selectivity. |
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Journal, issue, pages | Protein Sci., Vol. 8, Page 1455-1462, Year 1999 |
Publish date | Feb 3, 1999 (structure data deposition date) |
Authors | Pavlovsky, A.G. / Williams, M.G. / Ye, Q.Z. / Ortwine, D.F. / Purchase II, C.F. / White, A.D. / Dhanaraj, V. / Roth, B.D. / Johnson, L.L. / Hupe, D. ...Pavlovsky, A.G. / Williams, M.G. / Ye, Q.Z. / Ortwine, D.F. / Purchase II, C.F. / White, A.D. / Dhanaraj, V. / Roth, B.D. / Johnson, L.L. / Hupe, D. / Humblet, C. / Blundell, T.L. |
External links | PubMed:10422833 |
Methods | X-ray diffraction |
Resolution | 1.64 - 2 Å |
Structure data | PDB-1b8y: PDB-1caq: PDB-1ciz: PDB-1qia: PDB-1qic: |
Chemicals | ChemComp-ZN: ChemComp-CA: ChemComp-SO4: ChemComp-IN7: ChemComp-HOH: ChemComp-DPS: |
Source |
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Keywords | HYDROLASE / MATRIX METALLOPROTEINASE-3 / STROMELYSIN-1 / MATRIX METALLOPROTEINASE / MMP-3 / NON-PEPTIDE INHIBITOR / METALLOPROTEINASE / INHIBITOR / MATRIXIN / MATRIX METALLOPROTEINASE-3 (MMP-3) / METZINCIN |