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-Structure paper
Title | Crystal structure of human proto-oncogene serine threonine kinase (PIM1) in complex with a consensus peptide and a furan-thiazolidinedione ligand |
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Journal, issue, pages | To be Published |
Publish date | Jan 21, 2011 (structure data deposition date) |
Authors | Filippakopoulos, P. / Bullock, A.N. / Fedorov, O. / Miduturu, C.V. / von Delft, F. / Arrowsmith, C.H. / Weigelt, J. / Edwards, A. / Bountra, C. / Grey, N. ...Filippakopoulos, P. / Bullock, A.N. / Fedorov, O. / Miduturu, C.V. / von Delft, F. / Arrowsmith, C.H. / Weigelt, J. / Edwards, A. / Bountra, C. / Grey, N. / Knapp, S. / Structural Genomics Consortium (SGC) |
External links | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | PDB-3qf9: |
Chemicals | ChemComp-NM8: ChemComp-NA: ChemComp-CL: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE/PEPTIDE / COMPLEX TRANSFERASE-PEPTIDE / PIM1 / KINASE / CANCER / LEUKEMIA / ATP-BINDING / NUCLEAR PROTEIN / NUCLEOTIDE-BINDING / PHOSPHORYLATION / PROTO-ONCOGENE / SERINE/THREONINE-PROTEIN KINASE / TRANSFERASE / Structural Genomics Consortium / SGC / TRANSFERASE-TRANSFERASE INHIBITOR complex |