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-Structure paper
Title | A small molecule VHL molecular glue degrader for cysteine dioxygenase 1 |
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Journal, issue, pages | To Be Published |
Publish date | Jan 11, 2024 (structure data deposition date) |
![]() | Tutter, A. / Buckley, D. / Golosov, A. / Ma, X. / Shu, W. / Michaud, G. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.5 - 2.9 Å |
Structure data | ![]() PDB-8vl9: ![]() PDB-8vlb: |
Chemicals | ![]() PDB-1aci: ![]() ChemComp-CIT: ![]() ChemComp-FE2: ![]() ChemComp-HOH: ![]() ChemComp-3JF: |
Source |
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![]() | APOPTOSIS / VHL / CDO1 / VHL-small molecule-CDO1 ternary complex / degradation |