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-Structure paper
Title | Structural Basis for DCAF2 as a Novel E3 Ligase for PROTAC-Mediated Targeted Protein Degradation |
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Journal, issue, pages | Structure, Year 2025 |
Publish date | Jun 6, 2024 (structure data deposition date) |
![]() | McMahon EJ / Cioffi AG / Visperas PR / Lin Y / Shaghafi M / Daczkowski CM / Hermann JC / Everley RA / Neve RM / Erlanson DA ...McMahon EJ / Cioffi AG / Visperas PR / Lin Y / Shaghafi M / Daczkowski CM / Hermann JC / Everley RA / Neve RM / Erlanson DA / Webster KR / Narayan V / Wang W |
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Methods | EM (single particle) |
Resolution | 3.05 - 3.36 Å |
Structure data | EMDB-45224, PDB-9c5t: EMDB-45225, PDB-9c5u: EMDB-45226, PDB-9c5v: |
Chemicals | ![]() PDB-1aum: ![]() PDB-1auo: |
Source |
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![]() | LIGASE / DCAF2 / E3 ligase / DTL / DDB1 / covalent / fragment / DDA1 / BRD4 / degrader |