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Title | A novel CLK inhibitor exhibits anti-tumor efficacies via modulating pre-mRNA splicing and targeting a MYC-dependent vulnerability |
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Journal, issue, pages | Embo Mol Med, Year 2018 |
Publish date | Jan 31, 2017 (structure data deposition date) |
![]() | Iwai, K. / Yaguchi, M. / Klein, M.G. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.92 Å |
Structure data | ![]() PDB-5unp: |
Chemicals | ![]() ChemComp-8FY: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / Protein Kinase / Dual Specificity Protein Kinase / Inhibitor / Transferase / complex / TRANSFERASE-TRANSFERASE INHIBITOR complex |