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Title | Discovery and Optimization of Small-Molecule Inhibitors for the BPTF Bromodomains Proteins |
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Journal, issue, pages | To Be Published |
Publish date | Jan 25, 2020 (structure data deposition date) |
![]() | Lu, T. / Lu, H.B. / Wang, J. / Han, J. / Xiao, S. / Jiang, H. / Chen, Y. / Yang, F. / Li, Q. / Jiang, H.L. ...Lu, T. / Lu, H.B. / Wang, J. / Han, J. / Xiao, S. / Jiang, H. / Chen, Y. / Yang, F. / Li, Q. / Jiang, H.L. / Chen, K.X. / Lu, W.C. / Lin, H. / Luo, C. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.5715086186 - 2.20017124371 Å |
Structure data | ![]() PDB-6lu5: ![]() PDB-6lu6: ![]() PDB-7f5c: ![]() PDB-7f5d: ![]() PDB-7f5e: |
Chemicals | ![]() ChemComp-EUO: ![]() ChemComp-HOH: ![]() ChemComp-EUU: ![]() ChemComp-1IY: |
Source |
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![]() | ANTITUMOR PROTEIN / BPTF Bromodomain / Lysine acetylation / small-molecule inhibitor / high-throughput screening / BIOSYNTHETIC PROTEIN |