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-Structure paper
Title | Allosteric Inhibitors of VAV1 Block Guanine Nucleotide Exchange Activity |
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Journal, issue, pages | To Be Published |
Publish date | Dec 18, 2018 (structure data deposition date) |
![]() | Gerspacher, M. / Skaanderup, P.R. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.5 - 2.7 Å |
Structure data | ![]() PDB-6new: ![]() PDB-6nf1: ![]() PDB-6nfa: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-HOH: ![]() ChemComp-9JY: ![]() ChemComp-MES: ![]() ChemComp-9K1: |
Source |
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![]() | METAL BINDING PROTEIN / GEF / Rac / Vav1 / METAL BINDING PROTEIN/INHIBITOR / inhibitor / METAL BINDING PROTEIN-INHIBITOR complex / SIGNALING PROTEIN/INHIBITOR / SIGNALING PROTEIN-INHIBITOR complex |