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-Structure paper
Title | The PDE inhibition profile of LY294002 and tetrahydropyranyl analogues reveals a chromone motif for the development of PDE inhibitors |
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Journal, issue, pages | To be Published |
Publish date | Jan 15, 2014 (structure data deposition date) |
![]() | Howard, B.L. / Nankervis, J.L. / Feil, S.C. / Manallack, D.T. / Holien, J.K. / Zhen, Z. / Jennings, I.G. / Abbott, B.M. / Parker, M.W. / Thompson, P.E. |
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Methods | X-ray diffraction |
Resolution | 2.032 Å |
Structure data | ![]() PDB-4ogb: |
Chemicals | ![]() ChemComp-2SR: ![]() ChemComp-EDO: ![]() ChemComp-PEG: ![]() ChemComp-ZN: ![]() ChemComp-DMS: ![]() ChemComp-EPE: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / CATALYTIC MECHANISM / CAMP HYDROLYSIS / HYDROLASE-INHIBITOR COMPLEX / HYDROLASE-HYDROLASE INHIBITOR complex |