| タイトル | Creating a Resistance Model for TGT: The Effect of Mutations on Flexible lin-Benzoguanine Substituents | 
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| ジャーナル・号・ページ | To be Published | 
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| 掲載日 | 2014年4月28日 (構造データの登録日) | 
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|  著者 | Neeb, M. / Heine, A. / Klebe, G. | 
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|  リンク | PubMedで検索 | 
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| 手法 | X線回折 | 
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| 解像度 | 1.241 - 1.887 Å | 
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| 構造データ | PDB-4q8m: tRNA-Guanine Transglycosylase (TGT) Mutant V262T Apo Structure
 手法: X-RAY DIFFRACTION / 解像度: 1.241 Å
PDB-4q8n: tRNA-Guanine Transglycosylase (TGT) Mutant V262C Apo Structure
 手法: X-RAY DIFFRACTION / 解像度: 1.449 Å
PDB-4q8o: tRNA-Guanine Transglycosylase (TGT) Mutant V262T in Complex with 6-Amino-2-{[2-(morpholin-4-yl)ethyl]amino}-1H,7H,8H-imidazo[4,5-g]quinazolin-8-one
 手法: X-RAY DIFFRACTION / 解像度: 1.887 Å
PDB-4q8p: tRNA-Guanine Transglycosylase (TGT) Mutant V262D in Complex with 6-Amino-2-{[2-(morpholin-4-yl)ethyl]amino}-1H,7H,8H-imidazo[4,5-g]quinazolin-8-one
 手法: X-RAY DIFFRACTION / 解像度: 1.45 Å
PDB-4q8q: tRNA-Guanine Transglycosylase (TGT) Mutant V262C in Complex with 6-Amino-2-{[2-(morpholin-4-yl)ethyl]amino}-1H,7H,8H-imidazo[4,5-g]quinazolin-8-one
 手法: X-RAY DIFFRACTION / 解像度: 1.721 Å
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| 化合物 | ChemComp-CKR: 6-amino-2-[(2-morpholin-4-ylethyl)amino]-3,7-dihydro-8H-imidazo[4,5-g]quinazolin-8-one
 
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| 由来 |  zymomonas mobilis subsp. mobilis (バクテリア)
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|  キーワード | Transferase/transferase inhibitor / preQ1 / tRNA / Transferase-transferase inhibitor complex / Guanine Exchange Enzyme / Transferase | 
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