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-Structure paper
| Title | Discovery of ART5537: A Potent and Selective Small-Molecule Probe for EXO1. |
|---|---|
| Journal, issue, pages | J. Med. Chem., Vol. 68, Page 26432-26447, Year 2025 |
| Publish date | Aug 15, 2025 (structure data deposition date) |
Authors | Mann, S.E. / Davis, O.A. / Bomke, J. / Cornaciu, I. / Elinati, E. / Follows, B. / Galbiati, A. / Geo, L. / Grande, D. / Jorand-Lebrun, C. ...Mann, S.E. / Davis, O.A. / Bomke, J. / Cornaciu, I. / Elinati, E. / Follows, B. / Galbiati, A. / Geo, L. / Grande, D. / Jorand-Lebrun, C. / Lademann, C.A. / Lefranc, J. / Leuthner, B. / Mason, B. / McWhirter, C.L. / Musil, D. / Pehl, U. / Petersson, C. / Pica, A. / Pinto, M.F. / Rajendra, E. / Rakers, C. / Rego, A.T. / Robinson, H.M.R. / Schwarz, D. / Smith, G.C.M. / Sorrell, F.J. / Zenke, F.T. / Heald, R.A. / Burgdorf, L.T. |
External links | J. Med. Chem. / PubMed:41359073 |
| Methods | X-ray diffraction |
| Resolution | 1.9 - 2.199 Å |
| Structure data | ![]() PDB-9seb: ![]() PDB-9smo: |
| Chemicals | ![]() ChemComp-MG: ![]() ChemComp-NA: ![]()
PDB-1jnc: Unknown entry ![]() ChemComp-FMT: ![]() ChemComp-HOH: ![]() PDB-1jo0: |
| Source |
|
Keywords | HYDROLASE / Exonuclease |
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