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| Title | Potent and selective SETDB1 covalent negative allosteric modulator reduces methyltransferase activity in cells. |
|---|---|
| Journal, issue, pages | Nat Commun, Vol. 16, Page 1905-1905, Year 2025 |
| Publish date | Jul 26, 2024 (structure data deposition date) |
Authors | Uguen, M. / Shell, D.J. / Silva, M. / Deng, Y. / Li, F. / Szewczyk, M.M. / Yang, K. / Zhao, Y. / Stashko, M.A. / Norris-Drouin, J.L. ...Uguen, M. / Shell, D.J. / Silva, M. / Deng, Y. / Li, F. / Szewczyk, M.M. / Yang, K. / Zhao, Y. / Stashko, M.A. / Norris-Drouin, J.L. / Waybright, J.M. / Beldar, S. / Rectenwald, J.M. / Mordant, A.L. / Webb, T.S. / Herring, L.E. / Arrowsmith, C.H. / Ackloo, S. / Gygi, S.P. / McGinty, R.K. / Barsyte-Lovejoy, D. / Liu, P. / Halabelian, L. / James, L.I. / Pearce, K.H. / Frye, S.V. |
External links | Nat Commun / PubMed:39994194 |
| Methods | X-ray diffraction |
| Resolution | 1.27 - 1.53 Å |
| Structure data | ![]() PDB-9cuw: ![]() PDB-9cux: |
| Chemicals | ![]() PDB-1az6: ![]() ChemComp-EDO: ![]() ChemComp-UNX: ![]() ChemComp-HOH: ![]() PDB-1az5: ![]() ChemComp-SO4: |
| Source |
|
Keywords | TRANSFERASE / Tudor domain / SETDB1 / SGC |
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