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| Title | Nonsymmetrically Substituted 1,1'-Biphenyl-Based Small Molecule Inhibitors of the PD-1/PD-L1 Interaction. |
|---|---|
| Journal, issue, pages | Acs Med. Chem. Lett., Vol. 15, Page 828-836, Year 2024 |
| Publish date | Mar 14, 2024 (structure data deposition date) |
Authors | Hec-Galazka, A. / Tyrcha, U. / Barczynski, J. / Bielski, P. / Mikitiuk, M. / Gudz, G.P. / Kitel, R. / Musielak, B. / Plewka, J. / Sitar, T. / Holak, T.A. |
External links | Acs Med. Chem. Lett. / PubMed:38894909 |
| Methods | X-ray diffraction |
| Resolution | 2.5 Å |
| Structure data | ![]() PDB-9eo0: |
| Chemicals | ![]() PDB-1h56: ![]() ChemComp-SO4: ![]() ChemComp-HOH: |
| Source |
|
Keywords | ANTITUMOR PROTEIN / PD-L1 / SMI / Nonsymmetrically |
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