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Title | Redirecting raltitrexed from cancer cell thymidylate synthase to Mycobacterium tuberculosis phosphopantetheinyl transferase. |
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Journal, issue, pages | Sci Adv, Vol. 10, Page eadj6406-eadj6406, Year 2024 |
Publish date | Mar 18, 2023 (structure data deposition date) |
Authors | Singh, A. / Ottavi, S. / Krieger, I. / Planck, K. / Perkowski, A. / Kaneko, T. / Davis, A.M. / Suh, C. / Zhang, D. / Goullieux, L. ...Singh, A. / Ottavi, S. / Krieger, I. / Planck, K. / Perkowski, A. / Kaneko, T. / Davis, A.M. / Suh, C. / Zhang, D. / Goullieux, L. / Alex, A. / Roubert, C. / Gardner, M. / Preston, M. / Smith, D.M. / Ling, Y. / Roberts, J. / Cautain, B. / Upton, A. / Cooper, C.B. / Serbina, N. / Tanvir, Z. / Mosior, J. / Ouerfelli, O. / Yang, G. / Gold, B.S. / Rhee, K.Y. / Sacchettini, J.C. / Fotouhi, N. / Aube, J. / Nathan, C. |
External links | Sci Adv / PubMed:38489355 |
Methods | X-ray diffraction |
Resolution | 2.45 Å |
Structure data | PDB-8gkf: |
Chemicals | ChemComp-D16: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / complex / inhibitor / drug / Structural Genomics / TB Structural Genomics Consortium / TBSGC |