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-Structure paper
Title | Discovery of a cystathionine gamma-lyase (CSE) selective inhibitor targeting active-site pyridoxal 5'-phosphate (PLP) via Schiff base formation. |
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Journal, issue, pages | Sci Rep, Vol. 13, Page 16456-16456, Year 2023 |
Publish date | Apr 26, 2023 (structure data deposition date) |
Authors | Echizen, H. / Hanaoka, K. / Shimamoto, K. / Hibi, R. / Toma-Fukai, S. / Ohno, H. / Sasaki, E. / Komatsu, T. / Ueno, T. / Tsuchiya, Y. ...Echizen, H. / Hanaoka, K. / Shimamoto, K. / Hibi, R. / Toma-Fukai, S. / Ohno, H. / Sasaki, E. / Komatsu, T. / Ueno, T. / Tsuchiya, Y. / Watanabe, Y. / Otsuka, T. / Saito, H. / Nagatoishi, S. / Tsumoto, K. / Kojima, H. / Okabe, T. / Shimizu, T. / Urano, Y. |
External links | Sci Rep / PubMed:37777556 |
Methods | X-ray diffraction |
Resolution | 1.9 Å |
Structure data | PDB-8j6n: |
Chemicals |
ChemComp-TVJ: ChemComp-GOL: ChemComp-EDO: ChemComp-HOH: |
Source |
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Keywords | LYASE |