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-Structure paper
Title | Discovery of quinazoline HPK1 inhibitors with high cellular potency. |
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Journal, issue, pages | Bioorg. Med. Chem., Vol. 92, Page 117423-117423, Year 2023 |
Publish date | Feb 1, 2023 (structure data deposition date) |
![]() | Toure, M. / Johnson, T. / Li, B. / Schmidt, R. / Ma, H. / Neagu, C. / Lopez, A.U. / Wang, Y. / Guler, S. / Xiao, Y. ...Toure, M. / Johnson, T. / Li, B. / Schmidt, R. / Ma, H. / Neagu, C. / Lopez, A.U. / Wang, Y. / Guler, S. / Xiao, Y. / Henkes, R. / Ho, K. / Zhang, S. / Chu, C.L. / Gundra, U.M. / Porichis, F. / Li, L. / Maurer, C.K. / Fang, Z. / Musil, D. / DiPoto, M. / Friis, E. / Jones, R. / Jones, C. / Cummings, J. / Chekler, E. / Tanzer, E.M. / Huck, B. / Sherer, B. |
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Methods | X-ray diffraction |
Resolution | 1.941 - 2.821 Å |
Structure data | ![]() PDB-8cdw: ![]() PDB-8cij: |
Chemicals | ![]() ChemComp-UES: ![]() ChemComp-HOH: ![]() ChemComp-USF: |
Source |
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![]() | TRANSFERASE / PROTEIN KINASE / SIGNALING PROTEIN / MAP4K1 / HEMATOPOIETIC PROGENITOR KINASE |