| タイトル | Engineering broad-spectrum inhibitors of inflammatory chemokines from subclass A3 tick evasins. |
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| ジャーナル・号・ページ | Nat Commun, Vol. 14, Page 4204-4204, Year 2023 |
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| 掲載日 | 2021年9月29日 (構造データの登録日) |
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著者 | Devkota, S.R. / Aryal, P. / Pokhrel, R. / Jiao, W. / Perry, A. / Panjikar, S. / Payne, R.J. / Wilce, M.C.J. / Bhusal, R.P. / Stone, M.J. |
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リンク | Nat Commun / PubMed:37452046 |
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| 手法 | X線回折 |
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| 解像度 | 1.51 - 2.91 Å |
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| 構造データ | PDB-7scs: Crystal Structure of the Tick Evasin EVA-AAM1001 Complexed to Human Chemokine CCL11 手法: X-RAY DIFFRACTION / 解像度: 1.51 Å PDB-7sct: Crystal Structure of the Tick Evasin EVA-AAM1001 Complexed to Human Chemokine CCL16 手法: X-RAY DIFFRACTION / 解像度: 1.84 Å PDB-7scv: Crystal Structure of the Tick Evasin EVA-AAM1001 Complexed to Human Chemokine CCL17 手法: X-RAY DIFFRACTION / 解像度: 2.01 Å PDB-8fj0: Crystal Structure of the Tick Evasin EVA-AAM1001(Y44A) Complexed to Human Chemokine CCL2 手法: X-RAY DIFFRACTION / 解像度: 2.91 Å PDB-8fj2: Crystal Structure of the Tick Evasin EVA-AAM1001(C8) Complexed to Human Chemokine CCL17 手法: X-RAY DIFFRACTION / 解像度: 2.07 Å PDB-8fj3: Crystal Structure of the Tick Evasin EVA-AAM1001 Complexed to Human Chemokine CCL7(Y13A) 手法: X-RAY DIFFRACTION / 解像度: 2.07 Å PDB-8fk6: Crystal Structure of the Tick Evasin EVA-AAM1001(Y44A) Complexed to Human Chemokine CCL7 手法: X-RAY DIFFRACTION / 解像度: 1.74 Å PDB-8fk8: Crystal Structure of the Tick Evasin EVA-AAM1001(L39P) Complexed to Human Chemokine CCL7 手法: X-RAY DIFFRACTION / 解像度: 1.96 Å |
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| 化合物 | |
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| 由来 | amblyomma americanum (ダニ) homo sapiens (ヒト)
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キーワード | IMMUNE SYSTEM / Chemokine / Evasin / Ticks / Inflammation / Evasins / CYTOKINE / Tick / Anti-inflammatory / Chemokine-binding protein |
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