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| Title | Crystal structure of active CDK4-cyclin D and mechanistic basis for abemaciclib efficacy. |
|---|---|
| Journal, issue, pages | NPJ Breast Cancer, Vol. 8, Page 126-126, Year 2022 |
| Publish date | Oct 15, 2021 (structure data deposition date) |
Authors | Gharbi, S.I. / Pelletier, L.A. / Espada, A. / Gutierrez, J. / Sanfeliciano, S.M.G. / Rauch, C.T. / Ganado, M.P. / Baquero, C. / Zapatero, E. / Zhang, A. ...Gharbi, S.I. / Pelletier, L.A. / Espada, A. / Gutierrez, J. / Sanfeliciano, S.M.G. / Rauch, C.T. / Ganado, M.P. / Baquero, C. / Zapatero, E. / Zhang, A. / Benach, J. / Russell, A.M. / Cano, L. / Gomez, S. / Broughton, H. / Pulliam, N. / Perez, C.M. / Torres, R. / Debets, M.F. / de Dios, A. / Puig, O. / Hilgers, M.T. / Lallena, M.J. |
External links | NPJ Breast Cancer / PubMed:36446794 |
| Methods | X-ray diffraction |
| Resolution | 2.51 Å |
| Structure data | ![]() PDB-7sj3: |
| Chemicals | ![]() ChemComp-6ZV: ![]() ChemComp-HOH: |
| Source |
|
Keywords | CELL CYCLE / CDK / cyclin / kinase / inhibitor complex |
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homo sapiens (human)
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