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-Structure paper
Title | Inhibiting ACK1-mediated phosphorylation of C-terminal Src kinase counteracts prostate cancer immune checkpoint blockade resistance. |
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Journal, issue, pages | Nat Commun, Vol. 13, Page 6929-6929, Year 2022 |
Publish date | Nov 10, 2020 (structure data deposition date) |
![]() | Sridaran, D. / Chouhan, S. / Mahajan, K. / Renganathan, A. / Weimholt, C. / Bhagwat, S. / Reimers, M. / Kim, E.H. / Thakur, M.K. / Saeed, M.A. ...Sridaran, D. / Chouhan, S. / Mahajan, K. / Renganathan, A. / Weimholt, C. / Bhagwat, S. / Reimers, M. / Kim, E.H. / Thakur, M.K. / Saeed, M.A. / Pachynski, R.K. / Seeliger, M.A. / Miller, W.T. / Feng, F.Y. / Mahajan, N.P. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.79 Å |
Structure data | ![]() PDB-7kp6: |
Chemicals | ![]() ChemComp-WTP: ![]() ChemComp-CL: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/INHIBITOR / protein-inhibitor complex / tyrosine kinase / TRANSFERASE / TRANSFERASE-INHIBITOR complex |