+Search query
-Structure paper
Title | Novel fragment-derived colchicine-site binders as microtubule-destabilizing agents. |
---|---|
Journal, issue, pages | Eur. J. Med. Chem., Vol. 241, Page 114614-114614, Year 2022 |
Publish date | Feb 28, 2022 (structure data deposition date) |
![]() | de la Roche, N.M. / Muhlethaler, T. / Di Martino, R.M.C. / Ortega, J.A. / Gioia, D. / Roy, B. / Prota, A.E. / Steinmetz, M.O. / Cavalli, A. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2 - 2.17 Å |
Structure data | ![]() PDB-7z2n: ![]() PDB-7z2p: |
Chemicals | ![]() ChemComp-GTP: ![]() ChemComp-MG: ![]() ChemComp-CA: ![]() ChemComp-GDP: ![]() ChemComp-MES: ![]() ChemComp-IAZ: ![]() ChemComp-ACP: ![]() ChemComp-HOH: ![]() ChemComp-NW6: |
Source |
|
![]() | CELL CYCLE / TUBULIN FOLD / CYTOSKELETON / MICROTUBULE |