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-Structure paper
Title | Cosolvent Sites-Based Discovery of Mycobacterium Tuberculosis Protein Kinase G Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 9691-9705, Year 2022 |
Publish date | Nov 2, 2021 (structure data deposition date) |
![]() | Burastero, O. / Defelipe, L.A. / Gola, G. / Tateosian, N.L. / Lopez, E.D. / Martinena, C.B. / Arcon, J.P. / Traian, M.D. / Wetzler, D.E. / Bento, I. ...Burastero, O. / Defelipe, L.A. / Gola, G. / Tateosian, N.L. / Lopez, E.D. / Martinena, C.B. / Arcon, J.P. / Traian, M.D. / Wetzler, D.E. / Bento, I. / Barril, X. / Ramirez, J. / Marti, M.A. / Garcia-Alai, M.M. / Turjanski, A.G. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.35 Å |
Structure data | ![]() PDB-7q52: |
Chemicals | ![]() ChemComp-FE: ![]() ChemComp-8ZC: ![]() ChemComp-NA: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / Tuberculosis / inhibitor / L2W |