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-Structure paper
Title | Development of Selective Phosphatidylinositol 5-Phosphate 4-Kinase gamma Inhibitors with a Non-ATP-competitive, Allosteric Binding Mode. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 3359-3370, Year 2022 |
Publish date | Dec 14, 2021 (structure data deposition date) |
Authors | Boffey, H.K. / Rooney, T.P.C. / Willems, H.M.G. / Edwards, S. / Green, C. / Howard, T. / Ogg, D. / Romero, T. / Scott, D.E. / Winpenny, D. ...Boffey, H.K. / Rooney, T.P.C. / Willems, H.M.G. / Edwards, S. / Green, C. / Howard, T. / Ogg, D. / Romero, T. / Scott, D.E. / Winpenny, D. / Duce, J. / Skidmore, J. / Clarke, J.H. / Andrews, S.P. |
External links | J. Med. Chem. / PubMed:35148092 |
Methods | X-ray diffraction |
Resolution | 1.95 - 2.39 Å |
Structure data | PDB-7qie: PDB-7qpn: |
Chemicals | ChemComp-DVF: ChemComp-HOH: ChemComp-ANP: |
Source |
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Keywords | TRANSFERASE / ALLOSTERIC BINDING / LIPID KINASE / NON-ATP-COMPETITIVE INHIBITOR / phosphatidylinositol 5-phosphate |