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-Structure paper
Title | From structure to clinic: Design of a muscarinic M1 receptor agonist with potential to treatment of Alzheimer's disease. |
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Journal, issue, pages | Cell, Vol. 184, Page 5886-, Year 2021 |
Publish date | Jun 18, 2020 (structure data deposition date) |
![]() | Brown, A.J.H. / Bradley, S.J. / Marshall, F.H. / Brown, G.A. / Bennett, K.A. / Brown, J. / Cansfield, J.E. / Cross, D.M. / de Graaf, C. / Hudson, B.D. ...Brown, A.J.H. / Bradley, S.J. / Marshall, F.H. / Brown, G.A. / Bennett, K.A. / Brown, J. / Cansfield, J.E. / Cross, D.M. / de Graaf, C. / Hudson, B.D. / Dwomoh, L. / Dias, J.M. / Errey, J.C. / Hurrell, E. / Liptrot, J. / Mattedi, G. / Molloy, C. / Nathan, P.J. / Okrasa, K. / Osborne, G. / Patel, J.C. / Pickworth, M. / Robertson, N. / Shahabi, S. / Bundgaard, C. / Phillips, K. / Broad, L.M. / Goonawardena, A.V. / Morairty, S.R. / Browning, M. / Perini, F. / Dawson, G.R. / Deakin, J.F.W. / Smith, R.T. / Sexton, P.M. / Warneck, J. / Vinson, M. / Tasker, T. / Tehan, B.G. / Teobald, B. / Christopoulos, A. / Langmead, C.J. / Jazayeri, A. / Cooke, R.M. / Rucktooa, P. / Congreve, M.S. / Weir, M. / Tobin, A.B. |
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Methods | X-ray diffraction |
Resolution | 2.17 - 2.5 Å |
Structure data | ![]() PDB-6zfz: ![]() PDB-6zg4: ![]() PDB-6zg9: |
Chemicals | ![]() ChemComp-QJT: ![]() ChemComp-OLA: ![]() ChemComp-PO4: ![]() ChemComp-OLC: ![]() ChemComp-EPE: ![]() ChemComp-PGE: ![]() ChemComp-HOH: ![]() ChemComp-QK8: ![]() ChemComp-QK2: |
Source |
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![]() | MEMBRANE PROTEIN / GPCR / 7TM |