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-Structure paper
Title | Macrocyclic Peptides as a Novel Class of NNMT Inhibitors: A SAR Study Aimed at Inhibitory Activity in the Cell. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 12, Page 1093-1101, Year 2021 |
Publish date | Mar 26, 2021 (structure data deposition date) |
Authors | Hayashi, K. / Uehara, S. / Yamamoto, S. / Cary, D.R. / Nishikawa, J. / Ueda, T. / Ozasa, H. / Mihara, K. / Yoshimura, N. / Kawai, T. ...Hayashi, K. / Uehara, S. / Yamamoto, S. / Cary, D.R. / Nishikawa, J. / Ueda, T. / Ozasa, H. / Mihara, K. / Yoshimura, N. / Kawai, T. / Ono, T. / Fumoto, M. / Mikamiyama, H. |
External links | Acs Med. Chem. Lett. / PubMed:34267879 |
Methods | X-ray diffraction |
Resolution | 1.9 - 2.5 Å |
Structure data | PDB-7egu: PDB-7ehz: PDB-7ei2: |
Chemicals | ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / Nicotinamide N-methyltransferase |