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-Structure paper
Title | Discovery of Diaminopyrimidine Carboxamide HPK1 Inhibitors as Preclinical Immunotherapy Tool Compounds. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 12, Page 653-661, Year 2021 |
Publish date | Mar 11, 2021 (structure data deposition date) |
Authors | Vara, B.A. / Levi, S.M. / Achab, A. / Candito, D.A. / Fradera, X. / Lesburg, C.A. / Kawamura, S. / Lacey, B.M. / Lim, J. / Methot, J.L. ...Vara, B.A. / Levi, S.M. / Achab, A. / Candito, D.A. / Fradera, X. / Lesburg, C.A. / Kawamura, S. / Lacey, B.M. / Lim, J. / Methot, J.L. / Xu, Z. / Xu, H. / Smith, D.M. / Piesvaux, J.A. / Miller, J.R. / Bittinger, M. / Ranganath, S.H. / Bennett, D.J. / DiMauro, E.F. / Pasternak, A. |
External links | Acs Med. Chem. Lett. / PubMed:33859804 |
Methods | X-ray diffraction |
Resolution | 1.93 - 2.43 Å |
Structure data | PDB-7m0k: PDB-7m0l: PDB-7m0m: |
Chemicals | ChemComp-YK7: ChemComp-HOH: ChemComp-YK4: ChemComp-YK1: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE inhibitor / HPK1 HEMATOPOIETIC PROGENITOR KINASE / TRANSFERASE / TRANSFERASE-TRANSFERASE inhibitor complex / TRANSFERASE/TRANSFERASE inhibiotr / TRANSFERASE-TRANSFERASE inhibiotr complex |