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-Structure paper
Title | Structural Basis of Prolyl Hydroxylase Domain Inhibition by Molidustat. |
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Journal, issue, pages | Chemmedchem, Vol. 16, Page 2082-2088, Year 2021 |
Publish date | Jun 8, 2020 (structure data deposition date) |
Authors | Figg Jr., W.D. / McDonough, M.A. / Chowdhury, R. / Nakashima, Y. / Zhang, Z. / Holt-Martyn, J.P. / Krajnc, A. / Schofield, C.J. |
External links | Chemmedchem / PubMed:33792169 |
Methods | X-ray diffraction |
Resolution | 1.79 - 2.01 Å |
Structure data | PDB-6zbn: PDB-6zbo: |
Chemicals | ChemComp-QEE: ChemComp-MN: ChemComp-GOL: ChemComp-HOH: ChemComp-QEQ: ChemComp-CL: |
Source |
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Keywords | OXIDOREDUCTASE / Inhibitor / Complex / IOX4 / HIF / PHD2 / Hypoxia / Molidustat |