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-Structure paper
Title | Structure Based Design of Bicyclic Peptide Inhibitors of RbAp48. |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 60, Page 1813-1820, Year 2021 |
Publish date | Jul 13, 2020 (structure data deposition date) |
Authors | Hart, P.'. / Hommen, P. / Noisier, A. / Krzyzanowski, A. / Schuler, D. / Porfetye, A.T. / Akbarzadeh, M. / Vetter, I.R. / Adihou, H. / Waldmann, H. |
External links | Angew. Chem. Int. Ed. Engl. / PubMed:33022847 |
Methods | X-ray diffraction |
Resolution | 2.5 - 2.6 Å |
Structure data | PDB-6zrc: PDB-6zrd: |
Chemicals | ChemComp-PXY: ChemComp-HOH: ChemComp-SEZ: |
Source |
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Keywords | CELL CYCLE / NURD / HISTONE BINDING DOMAIN / WD40 DOMAIN / BETA PROPELLER / CHROMATIN REGULATOR / MACROCYCLIC PEPTIDE |