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| Title | Structural Basis for alpha-Helix Mimicry and Inhibition of Protein-Protein Interactions with Oligourea Foldamers. |
|---|---|
| Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Year 2020 |
| Publish date | Aug 21, 2018 (structure data deposition date) |
Authors | Cussol, L. / Mauran-Ambrosino, L. / Buratto, J. / Belorusova, A.Y. / Neuville, M. / Osz, J. / Fribourg, S. / Fremaux, J. / Dolain, C. / Goudreau, S.R. ...Cussol, L. / Mauran-Ambrosino, L. / Buratto, J. / Belorusova, A.Y. / Neuville, M. / Osz, J. / Fribourg, S. / Fremaux, J. / Dolain, C. / Goudreau, S.R. / Rochel, N. / Guichard, G. |
External links | Angew. Chem. Int. Ed. Engl. / PubMed:32935897 |
| Methods | X-ray diffraction |
| Resolution | 1.79 - 2.372 Å |
| Structure data | ![]() PDB-6hfa: ![]() PDB-6xzh: ![]() PDB-6xzi: ![]() PDB-6xzj: ![]() PDB-6xzk: ![]() PDB-6xzv: |
| Chemicals | ![]() ChemComp-HOH: ![]() ChemComp-VDX: ![]() ChemComp-ACT: |
| Source |
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Keywords | ONCOPROTEIN / PROTEIN FOLDAMER COMPLEX / PROTEIN PROTEIN INTERACTION INHIBITOR / UREA BASED CHIMERA FOLDAMER / GENE REGULATION / Nuclear Receptor / Foldamer / Helix mimicry / Protein-protein Interaction |
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