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-Structure paper
Title | A Photoaffinity-Based Fragment-Screening Platform for Efficient Identification of Protein Ligands. |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 59, Page 21096-21105, Year 2020 |
Publish date | Sep 2, 2020 (structure data deposition date) |
Authors | Grant, E.K. / Fallon, D.J. / Hann, M.M. / Fantom, K.G.M. / Quinn, C. / Zappacosta, F. / Annan, R.S. / Chung, C.W. / Bamborough, P. / Dixon, D.P. ...Grant, E.K. / Fallon, D.J. / Hann, M.M. / Fantom, K.G.M. / Quinn, C. / Zappacosta, F. / Annan, R.S. / Chung, C.W. / Bamborough, P. / Dixon, D.P. / Stacey, P. / House, D. / Patel, V.K. / Tomkinson, N.C.O. / Bush, J.T. |
External links | Angew. Chem. Int. Ed. Engl. / PubMed:32745361 |
Methods | X-ray diffraction |
Resolution | 1.444 Å |
Structure data | PDB-7a9u: |
Chemicals | ChemComp-R5W: ChemComp-EDO: ChemComp-HOH: |
Source |
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Keywords | TRANSCRIPTION / INHIBITOR / HISTONE / EPIGENETIC READER / BROMODOMAIN / BRD4 / BROMODOMAIN CONTAINING PROTEIN 4 / ANTAGONIST |