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-Structure paper
Title | Discovery and Development of Small-Molecule Inhibitors of Glycogen Synthase. |
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Journal, issue, pages | J. Med. Chem., Vol. 63, Page 3538-3551, Year 2020 |
Publish date | Aug 31, 2019 (structure data deposition date) |
Authors | Tang, B. / Frasinyuk, M.S. / Chikwana, V.M. / Mahalingan, K.K. / Morgan, C.A. / Segvich, D.M. / Bondarenko, S.P. / Mrug, G.P. / Wyrebek, P. / Watt, D.S. ...Tang, B. / Frasinyuk, M.S. / Chikwana, V.M. / Mahalingan, K.K. / Morgan, C.A. / Segvich, D.M. / Bondarenko, S.P. / Mrug, G.P. / Wyrebek, P. / Watt, D.S. / DePaoli-Roach, A.A. / Roach, P.J. / Hurley, T.D. |
External links | J. Med. Chem. / PubMed:32134266 |
Methods | X-ray diffraction |
Resolution | 2.85 Å |
Structure data | PDB-6u77: |
Chemicals | ChemComp-G6P: ChemComp-VMC: |
Source |
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Keywords | TRANSFERASE/INHIBITOR / Inhibitor / Glycogen Synthase / TRANSFERASE / TRANSFERASE-INHIBITOR complex |