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-Structure paper
Title | Multicomponent Peptide Stapling as a Diversity-Driven Tool for the Development of Inhibitors of Protein-Protein Interactions. |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 59, Page 5235-5241, Year 2020 |
Publish date | Oct 8, 2019 (structure data deposition date) |
![]() | Ricardo, M.G. / Ali, A.M. / Plewka, J. / Surmiak, E. / Labuzek, B. / Neochoritis, C.G. / Atmaj, J. / Skalniak, L. / Zhang, R. / Holak, T.A. ...Ricardo, M.G. / Ali, A.M. / Plewka, J. / Surmiak, E. / Labuzek, B. / Neochoritis, C.G. / Atmaj, J. / Skalniak, L. / Zhang, R. / Holak, T.A. / Groves, M. / Rivera, D.G. / Domling, A. |
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Methods | X-ray diffraction |
Resolution | 1.8 - 2.4 Å |
Structure data | ![]() PDB-6t2d: ![]() PDB-6t2e: ![]() PDB-6t2f: |
Chemicals | ![]() ChemComp-EPE: ![]() ChemComp-DMS: ![]() ChemComp-M9E: ![]() ChemComp-HOH: ![]() ChemComp-M9H: |
Source |
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![]() | PEPTIDE BINDING PROTEIN / Inhibitor / Complex / MDM2 / Stapled peptides / Ugi MCR-based macrocyclizations |