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-Structure paper
Title | Structure-Guided Enhancement of Selectivity of Chemical Probe Inhibitors Targeting Bacterial Seryl-tRNA Synthetase. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 9703-9717, Year 2019 |
Publish date | Mar 14, 2019 (structure data deposition date) |
![]() | Cain, R. / Salimraj, R. / Punekar, A.S. / Bellini, D. / Fishwick, C.W.G. / Czaplewski, L. / Scott, D.J. / Harris, G. / Dowson, C.G. / Lloyd, A.J. / Roper, D.I. |
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Methods | X-ray diffraction |
Resolution | 1.5 - 2.6 Å |
Structure data | ![]() PDB-6r1m: ![]() PDB-6r1n: ![]() PDB-6r1o: |
Chemicals | ![]() ChemComp-SSA: ![]() ChemComp-PO4: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-PEG: ![]() ChemComp-MG: ![]() ChemComp-JPE: ![]() ChemComp-CL: ![]() ChemComp-SO4: ![]() ChemComp-DMS: ![]() ChemComp-TRS: |
Source |
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![]() | LIGASE / aminoacyl-tRNA synthetase / class II / protein synthesis / inhibitor |