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-Structure paper
Title | Structure-guided design of antibacterials that allosterically inhibit DNA gyrase. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 29, Page 1407-1412, Year 2019 |
Publish date | Mar 6, 2019 (structure data deposition date) |
![]() | Thalji, R.K. / Raha, K. / Andreotti, D. / Checchia, A. / Cui, H. / Meneghelli, G. / Profeta, R. / Tonelli, F. / Tommasi, S. / Bakshi, T. ...Thalji, R.K. / Raha, K. / Andreotti, D. / Checchia, A. / Cui, H. / Meneghelli, G. / Profeta, R. / Tonelli, F. / Tommasi, S. / Bakshi, T. / Donovan, B.T. / Howells, A. / Jain, S. / Nixon, C. / Quinque, G. / McCloskey, L. / Bax, B.D. / Neu, M. / Chan, P.F. / Stavenger, R.A. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.65 - 3.4 Å |
Structure data | ![]() PDB-6qx1: ![]() PDB-6qx2: |
Chemicals | ![]() ChemComp-MN: ![]() ChemComp-JK8: ![]() ChemComp-GOL: ![]() ChemComp-GLY: ![]() ChemComp-CL: ![]() ChemComp-HOH: |
Source |
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![]() | ISOMERASE / Inhibitor / DNA complex |