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-Structure paper
Title | PH-domain-binding inhibitors of nucleotide exchange factor BRAG2 disrupt Arf GTPase signaling. |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 15, Page 358-366, Year 2019 |
Publish date | Feb 3, 2018 (structure data deposition date) |
Authors | Nawrotek, A. / Benabdi, S. / Niyomchon, S. / Kryszke, M.H. / Ginestier, C. / Caneque, T. / Tepshi, L. / Mariani, A. / St Onge, R.P. / Giaever, G. ...Nawrotek, A. / Benabdi, S. / Niyomchon, S. / Kryszke, M.H. / Ginestier, C. / Caneque, T. / Tepshi, L. / Mariani, A. / St Onge, R.P. / Giaever, G. / Nislow, C. / Charafe-Jauffret, E. / Rodriguez, R. / Zeghouf, M. / Cherfils, J. |
External links | Nat. Chem. Biol. / PubMed:30742123 |
Methods | X-ray diffraction |
Resolution | 2.501 Å |
Structure data | PDB-6fne: |
Chemicals | ChemComp-DY5: ChemComp-2PE: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / ARF GEF |