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-Structure paper
Title | Discovery of Macrocyclic Inhibitors of Apurinic/Apyrimidinic Endonuclease 1. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 1971-1988, Year 2019 |
Publish date | Sep 24, 2018 (structure data deposition date) |
![]() | Trilles, R. / Beglov, D. / Chen, Q. / He, H. / Wireman, R. / Reed, A. / Chennamadhavuni, S. / Panek, J.S. / Brown, L.E. / Vajda, S. ...Trilles, R. / Beglov, D. / Chen, Q. / He, H. / Wireman, R. / Reed, A. / Chennamadhavuni, S. / Panek, J.S. / Brown, L.E. / Vajda, S. / Porco Jr., J.A. / Kelley, M.R. / Georgiadis, M.M. |
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Methods | X-ray diffraction |
Resolution | 1.442 - 2.09 Å |
Structure data | ![]() PDB-6mk3: ![]() PDB-6mkk: ![]() PDB-6mkm: ![]() PDB-6mko: |
Chemicals | ![]() ChemComp-DMS: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-MG: ![]() ChemComp-TRS: ![]() ChemComp-GOL: |
Source |
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![]() | LYASE / Apurinic/apyrimidinic endonuclease / DNA repair / abasic site / solvent mapping |