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Title | Small Molecules Co-targeting CKI alpha and the Transcriptional Kinases CDK7/9 Control AML in Preclinical Models. |
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Journal, issue, pages | Cell, Vol. 175, Page 171-185.e25, Year 2018 |
Publish date | Jul 3, 2018 (structure data deposition date) |
![]() | Minzel, W. / Venkatachalam, A. / Fink, A. / Hung, E. / Brachya, G. / Burstain, I. / Shaham, M. / Rivlin, A. / Omer, I. / Zinger, A. ...Minzel, W. / Venkatachalam, A. / Fink, A. / Hung, E. / Brachya, G. / Burstain, I. / Shaham, M. / Rivlin, A. / Omer, I. / Zinger, A. / Elias, S. / Winter, E. / Erdman, P.E. / Sullivan, R.W. / Fung, L. / Mercurio, F. / Li, D. / Vacca, J. / Kaushansky, N. / Shlush, L. / Oren, M. / Levine, R. / Pikarsky, E. / Snir-Alkalay, I. / Ben-Neriah, Y. |
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Methods | X-ray diffraction |
Resolution | 1.59 - 3.17 Å |
Structure data | ![]() PDB-6gzd: ![]() PDB-6gzh: ![]() PDB-6gzm: |
Chemicals | ![]() ChemComp-DMS: ![]() ChemComp-PGE: ![]() ChemComp-EDO: ![]() ChemComp-PEG: ![]() ChemComp-TCE: ![]() ChemComp-LCI: ![]() ChemComp-HOH: ![]() ChemComp-GOL: ![]() ChemComp-CIT: |
Source |
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![]() | TRANSFERASE / CKIa / Casein kinase / Kinase inhibitor / CDK9 / A86 |