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-Structure paper
Title | Piperidinyl Ureas Chemically Control Defective in Cullin Neddylation 1 (DCN1)-Mediated Cullin Neddylation. |
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Journal, issue, pages | J. Med. Chem., Vol. 61, Page 2680-2693, Year 2018 |
Publish date | Oct 27, 2017 (structure data deposition date) |
Authors | Hammill, J.T. / Scott, D.C. / Min, J. / Connelly, M.C. / Holbrook, G. / Zhu, F. / Matheny, A. / Yang, L. / Singh, B. / Schulman, B.A. / Guy, R.K. |
External links | J. Med. Chem. / PubMed:29547696 |
Methods | X-ray diffraction |
Resolution | 1.05 - 1.1 Å |
Structure data | PDB-6bg3: PDB-6bg5: |
Chemicals | ChemComp-DOJ: ChemComp-HOH: ChemComp-DQD: |
Source |
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Keywords | HYDROLASE / LIGASE/INHIBITOR / E3 Ligase / LIGASE-INHIBITOR complex |