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-Structure paper
Title | Potent and Selective Inhibitors of Human Sirtuin 5. |
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Journal, issue, pages | J. Med. Chem., Vol. 61, Page 2460-2471, Year 2018 |
Publish date | Jan 25, 2018 (structure data deposition date) |
Authors | Kalbas, D. / Liebscher, S. / Nowak, T. / Meleshin, M. / Pannek, M. / Popp, C. / Alhalabi, Z. / Bordusa, F. / Sippl, W. / Steegborn, C. / Schutkowski, M. |
External links | J. Med. Chem. / PubMed:29494161 |
Methods | X-ray diffraction |
Resolution | 2.5 - 3.3 Å |
Structure data | PDB-6fky: PDB-6fkz: PDB-6flg: |
Chemicals | ChemComp-ZN: ChemComp-EPE: ChemComp-NA: ChemComp-EDO: ChemComp-E9N: ChemComp-DZK: ChemComp-HOH: ChemComp-GOL: ChemComp-DMS: |
Source |
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Keywords | SIGNALING PROTEIN / Sirtuin 5 / Inhibitor / Deacylase |