タイトル | CDKL Family Kinases Have Evolved Distinct Structural Features and Ciliary Function. |
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ジャーナル・号・ページ | Cell Rep, Vol. 22, Page 885-894, Year 2018 |
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掲載日 | 2012年11月30日 (構造データの登録日) |
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著者 | Canning, P. / Park, K. / Goncalves, J. / Li, C. / Howard, C.J. / Sharpe, T.D. / Holt, L.J. / Pelletier, L. / Bullock, A.N. / Leroux, M.R. |
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リンク | Cell Rep / PubMed:29420175 |
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手法 | X線回折 |
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解像度 | 1.53 - 2.4 Å |
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構造データ | PDB-3zdu: Crystal structure of the human CDKL3 kinase domain 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-4aaa: Crystal structure of the human CDKL2 kinase domain 手法: X-RAY DIFFRACTION / 解像度: 1.53 Å PDB-4agu: CRYSTAL STRUCTURE OF THE HUMAN CDKL1 KINASE DOMAIN 手法: X-RAY DIFFRACTION / 解像度: 2.4 Å PDB-4bbm: CRYSTAL STRUCTURE OF THE HUMAN CDKL2 KINASE DOMAIN WITH BOUND TCS 2312 手法: X-RAY DIFFRACTION / 解像度: 2 Å PDB-4bgq: Crystal structure of the human CDKL5 kinase domain 手法: X-RAY DIFFRACTION / 解像度: 2 Å |
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化合物 | ChemComp-38R: [4-({4-[(3-cyclopentyl-1H-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile
ChemComp-DKI: 5-AMINO-3-{[4-(AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4-TRIAZOLE-1-CARBOTHIOAMIDE
ChemComp-D15: N-(5-{[(2S)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1H-indazol-3-yl)benzamide
ChemComp-TC0: 4'-[5-[[3-[(CYCLOPROPYLAMINO)METHYL]PHENYL]AMINO]-1H-PYRAZOL-3-YL]-[1,1'-BIPHENYL]-2,4-DIOL
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由来 | - homo sapiens (ヒト)
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キーワード | TRANSFERASE / PHOSPHO-MIMETIC / KINASE |
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