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Title | New Insights into PI3K Inhibitor Design using X-ray Structures of PI3K alpha Complexed with a Potent Lead Compound. |
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Journal, issue, pages | Sci Rep, Vol. 7, Page 14572-14572, Year 2017 |
Publish date | Apr 13, 2017 (structure data deposition date) |
![]() | Yang, X. / Zhang, X. / Huang, M. / Song, K. / Li, X. / Meng, L. / Zhang, J. |
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Methods | X-ray diffraction |
Resolution | 2.97 Å |
Structure data | ![]() PDB-5xgh: |
Chemicals | ![]() ChemComp-84U: ![]() ChemComp-GOL: ![]() ChemComp-SO4: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/INHIBITOR / PI3K / inhibitor / TRANSFERASE-INHIBITOR complex |