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-Structure paper
Title | GNE-886: A Potent and Selective Inhibitor of the Cat Eye Syndrome Chromosome Region Candidate 2 Bromodomain (CECR2). |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 8, Page 737-741, Year 2017 |
Publish date | Mar 21, 2017 (structure data deposition date) |
![]() | Crawford, T.D. / Audia, J.E. / Bellon, S. / Burdick, D.J. / Bommi-Reddy, A. / Cote, A. / Cummings, R.T. / Duplessis, M. / Flynn, E.M. / Hewitt, M. ...Crawford, T.D. / Audia, J.E. / Bellon, S. / Burdick, D.J. / Bommi-Reddy, A. / Cote, A. / Cummings, R.T. / Duplessis, M. / Flynn, E.M. / Hewitt, M. / Huang, H.R. / Jayaram, H. / Jiang, Y. / Joshi, S. / Kiefer, J.R. / Murray, J. / Nasveschuk, C.G. / Neiss, A. / Pardo, E. / Romero, F.A. / Sandy, P. / Sims, R.J. / Tang, Y. / Taylor, A.M. / Tsui, V. / Wang, J. / Wang, S. / Wang, Y. / Xu, Z. / Zawadzke, L. / Zhu, X. / Albrecht, B.K. / Magnuson, S.R. / Cochran, A.G. |
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Methods | X-ray diffraction |
Resolution | 2.7 Å |
Structure data | ![]() PDB-5v84: |
Chemicals | ![]() ChemComp-SO4: ![]() ChemComp-96V: ![]() ChemComp-HOH: |
Source |
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![]() | Transcription/Inhibitor / Bromodomain / SBDD / Transcription-Inhibitor complex |