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-Structure paper
Title | Functional and structural analysis of AT-specific minor groove binders that disrupt DNA-protein interactions and cause disintegration of the Trypanosoma brucei kinetoplast. |
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Journal, issue, pages | Nucleic Acids Res., Vol. 45, Page 8378-8391, Year 2017 |
Publish date | Jul 15, 2016 (structure data deposition date) |
Authors | Millan, C.R. / Acosta-Reyes, F.J. / Lagartera, L. / Ebiloma, G.U. / Lemgruber, L. / Nue Martinez, J.J. / Saperas, N. / Dardonville, C. / de Koning, H.P. / Campos, J.L. |
External links | Nucleic Acids Res. / PubMed:28637278 |
Methods | X-ray diffraction |
Resolution | 1.25 - 1.43 Å |
Structure data | PDB-5lit: PDB-6gim: |
Chemicals | ChemComp-6XV: ChemComp-MG: ChemComp-HOH: ChemComp-EZK: |
Source |
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Keywords | DNA / All AT DNA / Antiparasitic Drug / Minor Groove Binding Drug / AT-rich DNA / DNA binding drugs / Minor groove binding drugs / antiparasitic drugs / Trypanosoma brucei |