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Title | Identification and Profiling of a Selective and Brain Penetrant Radioligand for in Vivo Target Occupancy Measurement of Casein Kinase 1 (CK1) Inhibitors. |
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Journal, issue, pages | ACS Chem Neurosci, Vol. 8, Page 1995-2004, Year 2017 |
Publish date | Jun 13, 2017 (structure data deposition date) |
![]() | Wager, T.T. / Galatsis, P. / Chandrasekaran, R.Y. / Butler, T.W. / Li, J. / Zhang, L. / Mente, S. / Subramanyam, C. / Liu, S. / Doran, A.C. ...Wager, T.T. / Galatsis, P. / Chandrasekaran, R.Y. / Butler, T.W. / Li, J. / Zhang, L. / Mente, S. / Subramanyam, C. / Liu, S. / Doran, A.C. / Chang, C. / Fisher, K. / Grimwood, S. / Hedde, J.R. / Marconi, M. / Schildknegt, K. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.99 Å |
Structure data | ![]() PDB-5w4w: |
Chemicals | ![]() ChemComp-9WG: ![]() ChemComp-SO4: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/INHIBITOR / kinase / inhibitor / TRANSFERASE-INHIBITOR complex |