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Title | Targeting S-adenosylmethionine biosynthesis with a novel allosteric inhibitor of Mat2A. |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 13, Page 785-792, Year 2017 |
Publish date | Jan 8, 2017 (structure data deposition date) |
Authors | Quinlan, C.L. / Kaiser, S.E. / Bolanos, B. / Nowlin, D. / Grantner, R. / Karlicek-Bryant, S. / Feng, J.L. / Jenkinson, S. / Freeman-Cook, K. / Dann, S.G. ...Quinlan, C.L. / Kaiser, S.E. / Bolanos, B. / Nowlin, D. / Grantner, R. / Karlicek-Bryant, S. / Feng, J.L. / Jenkinson, S. / Freeman-Cook, K. / Dann, S.G. / Wang, X. / Wells, P.A. / Fantin, V.R. / Stewart, A.E. / Grant, S.K. |
External links | Nat. Chem. Biol. / PubMed:28553945 |
Methods | X-ray diffraction |
Resolution | 2.062 Å |
Structure data | PDB-5ugh: |
Chemicals | ChemComp-8AJ: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / Mat2A / SAM / methionine adenosyltransferase |