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-Structure paper
Title | Thiophene antibacterials that allosterically stabilize DNA-cleavage complexes with DNA gyrase. |
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Journal, issue, pages | Proc. Natl. Acad. Sci. U.S.A., Vol. 114, Page E4492-E4500, Year 2017 |
Publish date | Apr 17, 2017 (structure data deposition date) |
![]() | Chan, P.F. / Germe, T. / Bax, B.D. / Huang, J. / Thalji, R.K. / Bacque, E. / Checchia, A. / Chen, D. / Cui, H. / Ding, X. ...Chan, P.F. / Germe, T. / Bax, B.D. / Huang, J. / Thalji, R.K. / Bacque, E. / Checchia, A. / Chen, D. / Cui, H. / Ding, X. / Ingraham, K. / McCloskey, L. / Raha, K. / Srikannathasan, V. / Maxwell, A. / Stavenger, R.A. |
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Methods | X-ray diffraction |
Resolution | 1.98 - 2.22 Å |
Structure data | ![]() PDB-5npk: ![]() PDB-5npp: |
Chemicals | ![]() ChemComp-MN: ![]() ChemComp-94H: ![]() ChemComp-GOL: ![]() ChemComp-CL: ![]() ChemComp-SO4: ![]() ChemComp-NA: ![]() ChemComp-9JN: ![]() ChemComp-HOH: ![]() ChemComp-94K: ![]() ChemComp-DMS: ![]() ChemComp-6EJ: |
Source |
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![]() | ISOMERASE / TYPE IIA TOPOISOMERASE / ANTIBACTERIAL / INHIBITOR |