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-Structure paper
Title | Ternary complex of human ROR gamma ligand-binding domain, inverse agonist and SMRT peptide shows a unique mechanism of corepressor recruitment |
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Journal, issue, pages | Genes Cells, Vol. 22, Page 535-551, Year 2017 |
Publish date | Mar 3, 2017 (structure data deposition date) |
Authors | Noguchi, M. / Nomura, A. / Murase, K. / Doi, S. / Yamaguchi, K. / Hirata, K. / Shiozaki, M. / Hirashima, S. / Kotoku, M. / Yamaguchi, T. ...Noguchi, M. / Nomura, A. / Murase, K. / Doi, S. / Yamaguchi, K. / Hirata, K. / Shiozaki, M. / Hirashima, S. / Kotoku, M. / Yamaguchi, T. / Katsuda, Y. / Steensma, R. / Li, X. / Tao, H. / Tse, B. / Fenn, M. / Babine, R. / Bradley, E. / Crowe, P. / Thacher, S. / Adachi, T. / Kamada, M. |
External links | Genes Cells / PubMed:28493531 |
Methods | X-ray diffraction |
Resolution | 2 - 2.6 Å |
Structure data | PDB-5x8q: PDB-5x8s: PDB-5x8u: PDB-5x8w: PDB-5x8x: |
Chemicals | ChemComp-82R: ChemComp-HOH: ChemComp-6Q5: ChemComp-82O: |
Source |
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Keywords | TRANSFERASE/IHIBITOR / Inhibitor / Ternary Complex / Nuclear Receptor / TRANSFERASE-IHIBITOR complex / TRANSFERASE/INHIBITOR / Binary Complex / TRANSFERASE-INHIBITOR complex / TRANSCRIPTION/INHIBITOR / TRANSCRIPTION-INHIBITOR complex |