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-Structure paper
Title | Structure-Based Design of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors Based on Paroxetine. |
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Journal, issue, pages | J. Med. Chem., Vol. 60, Page 3052-3069, Year 2017 |
Publish date | Jan 23, 2017 (structure data deposition date) |
Authors | Waldschmidt, H.V. / Homan, K.T. / Cato, M.C. / Cruz-Rodriguez, O. / Cannavo, A. / Wilson, M.W. / Song, J. / Cheung, J.Y. / Koch, W.J. / Tesmer, J.J. / Larsen, S.D. |
External links | J. Med. Chem. / PubMed:28323425 |
Methods | X-ray diffraction |
Resolution | 2.15 - 3.03 Å |
Structure data | PDB-5ukk: PDB-5ukl: PDB-5ukm: |
Chemicals | ChemComp-MG: ChemComp-8DJ: ChemComp-HOH: ChemComp-SIX: ChemComp-T0E: ChemComp-CMT: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / kinase / inhibitor complex / TRANSFERASE-TRANSFERASE INHIBITOR complex / Transferase/Signaling Protein / Transferase-Signaling Protein complex |