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-Structure paper
Title | Structure-based drug design of novel ASK1 inhibitors using an integrated lead optimization strategy. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 27, Page 1709-1713, Year 2017 |
Publish date | Mar 1, 2017 (structure data deposition date) |
![]() | Gibson, T.S. / Johnson, B. / Fanjul, A. / Halkowycz, P. / Dougan, D.R. / Cole, D. / Swann, S. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.5 - 3.1 Å |
Structure data | ![]() PDB-5v19: ![]() PDB-5v24: |
Chemicals | ![]() ChemComp-8V4: ![]() ChemComp-HOH: ![]() ChemComp-8V7: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE / METAL-BINDING / APOPTOSIS / TRANSFERASE-TRANSFERASE INHIBITOR complex |