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-Structure paper
Title | Design, Synthesis, and Cytotoxic Evaluation of Novel Tubulysin Analogues as ADC Payloads. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 7, Page 999-1004, Year 2016 |
Publish date | Jul 20, 2016 (structure data deposition date) |
Authors | Leverett, C.A. / Sukuru, S.C. / Vetelino, B.C. / Musto, S. / Parris, K. / Pandit, J. / Loganzo, F. / Varghese, A.H. / Bai, G. / Liu, B. ...Leverett, C.A. / Sukuru, S.C. / Vetelino, B.C. / Musto, S. / Parris, K. / Pandit, J. / Loganzo, F. / Varghese, A.H. / Bai, G. / Liu, B. / Liu, D. / Hudson, S. / Doppalapudi, V.R. / Stock, J. / O'Donnell, C.J. / Subramanyam, C. |
External links | ACS Med Chem Lett / PubMed:27882198 |
Methods | X-ray diffraction |
Resolution | 2.5 Å |
Structure data | PDB-5kx5: |
Chemicals | ChemComp-GTP: ChemComp-MG: ChemComp-CA: ChemComp-GDP: ChemComp-6YK: ChemComp-ADP: ChemComp-HOH: |
Source |
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Keywords | STRUCTURAL PROTEIN/INHIBITOR / Tubulin Tubulysin / STRUCTURAL PROTEIN-INHIBITOR complex |