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-Structure paper
Title | Selective Inhibition of Autotaxin Is Efficacious in Mouse Models of Liver Fibrosis. |
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Journal, issue, pages | J. Pharmacol. Exp. Ther., Vol. 360, Page 1-13, Year 2017 |
Publish date | Jul 20, 2016 (structure data deposition date) |
Authors | Bain, G. / Shannon, K.E. / Huang, F. / Darlington, J. / Goulet, L. / Prodanovich, P. / Ma, G.L. / Santini, A.M. / Stein, A.J. / Lonergan, D. ...Bain, G. / Shannon, K.E. / Huang, F. / Darlington, J. / Goulet, L. / Prodanovich, P. / Ma, G.L. / Santini, A.M. / Stein, A.J. / Lonergan, D. / King, C.D. / Calderon, I. / Lai, A. / Hutchinson, J.H. / Evans, J.F. |
External links | J. Pharmacol. Exp. Ther. / PubMed:27754931 |
Methods | X-ray diffraction |
Resolution | 2.59 Å |
Structure data | PDB-5kxa: |
Chemicals | ChemComp-NAG: ChemComp-ZN: ChemComp-CA: ChemComp-6Y7: ChemComp-PO4: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE/HYDROLASE INHIBITOR / ENPP2 / autotaxin / HYDROLASE-HYDROLASE INHIBITOR complex |